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Molfinity

GLP-1R Antagonist 1 - CAS 488097-06-9

GLP-1R Antagonist 1 - CAS 488097-06-9

SKU:MF-0012429-01

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  • Bioactivity

    GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM) .

  • Target

    Glucagon Receptor

  • Related Pathways

    GPCR/G Protein

  • CAS Number

    488097-06-9

  • Purity

    0.9984

  • Molecular Formula

    C16H11ClF6N4O2

  • Molecular Weight

    440.73

  • SMILES

    Cn1c2NC(=NC(c2c(=O)n(C)c1=O)(C(F)(F)F)C(F)(F)F)c1ccc(Cl)cc1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound