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GLP-1R Antagonist 1 - CAS 488097-06-9
GLP-1R Antagonist 1 - CAS 488097-06-9
SKU:MF-0012429-01
Regular price
$38.41 USD
Regular price
$24.70 USD
Sale price
$38.41 USD
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Product Details
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Bioactivity
GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM) .
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Target
Glucagon Receptor
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Related Pathways
GPCR/G Protein
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CAS Number
488097-06-9
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Purity
0.9984
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Molecular Formula
C16H11ClF6N4O2
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Molecular Weight
440.73
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SMILES
Cn1c2NC(=NC(c2c(=O)n(C)c1=O)(C(F)(F)F)C(F)(F)F)c1ccc(Cl)cc1
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Storage Temperature
-20°C
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Shipping Conditions
Ice Packs
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Category
Small Compound