Glucocorticoid receptor-IN-1 - CAS 2662908-25-8

Glucocorticoid receptor-IN-1 is a selective regulator of the glucocorticoid receptor (GR) and exhibits anti-inflammatory activity. glucocorticoid receptor-IN-1 has good transcriptional repression, acting on hMMP1 (IC50: 2.11 nM) and also has a transcriptional activating effect on MMTV (EC50: 5.59 nM) .

Others, Glucocorticoid Receptor, MMP

Endocrinology/Hormones, Proteases/Proteasome, Others

2662875

C24H19F4N7O2

513.45

O([C@@H]([C@@H](NC(C(C)(F)F)=O)C)C1=CC(F)=CC(F)=C1)C=2C=C3C(N(N=N3)C4=CN5C(C=C4)=NN=C5)=CC2

-20°C

Ice Packs

Small Compound