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Molfinity

GNE-207 - CAS 2158266-58-9

GNE-207 - CAS 2158266-58-9

MF-0032931-01

$1,910.30 USD
$1,910.30 USD
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Product Details

  • Bioactivity

    GNE-207 is a selective and orally bioavailable inhibitor of the bromodomain of CBP (IC50: 1 nM) . It has a selective index of >2500-fold against BRD4 (1) . GNE-207 displays excellent CBP potency (EC50: 18 nM for MYC expression in MV-4-11 cells) .

  • Target

    Histone Acetyltransferase, Epigenetic Reader Domain

  • Related Pathways

    Chromatin/Epigenetic

  • CAS Number

    2158199

  • Molecular Formula

    C29H30N6O3

  • Molecular Weight

    510.59

  • SMILES

    CNC(=O)c1ccc(cn1)-c1cc2cccc(-c3nn(C4CCOCC4)c4CCN(Cc34)C(C)=O)c2cn1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound