GPS1573 - CAS 2445822-54-6

GPS1573 is a non-competitive antagonist of the melanocortin 2 receptor (MC2R) that blocks the ACTH-stimulated activity of MC2R in a dose-dependent manner (IC50=66 nM) . Due to its high selectivity in antagonizing MC2R, GPS1573 is utilized for research in Cushings disease.

2445822-54-6

C86H138N28O14

1788.19

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-20°C

Ice Packs

Small Compound