GR 64349 - CAS 137593-52-3

Potent and selective tachykinin NK2 receptor agonist (EC50 = 3.7 nM in rat colon) . Displays > 1000- and > 300-fold selectivity over NK1 and NK3 receptors respectively. Active in vivo.

Neurokinin receptor

Neuroscience, GPCR/G Protein

137538

C42H68N10O11S

921.12

CSCC[C@H](NC(=O)[C@H](CC(C)C)N1CC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CO)NC(=O)[C@H](CC(O)=O)NC(=O)[C@@H](N)CCCCN)C(C)C)C1=O)C(N)=O

-20°C

Ice Packs

Peptide