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GRK2 Inhibitor 2 - CAS 2592436-21-8

GRK2 Inhibitor 2 - CAS 2592436-21-8

MF-0157540-01

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Product Details

  • Bioactivity

    GRK2 Inhibitor 2 (Compound 8h), with an IC50 of 19 nM for GRK2 and 137 nM for Aurora-A, enhances β-AR-mediated cAMP accumulation in GRK2-overexpressing HEK293 cells. It is utilized in congestive heart failure (HF) research [1].

  • Target

    Aurora Kinase, Others, GRK

  • Related Pathways

    Cell Cycle/Checkpoint, GPCR/G Protein, Others, Chromatin/Epigenetic

  • CAS Number

    2592407

  • Molecular Formula

    C19H16N4O2

  • Molecular Weight

    332.36

  • SMILES

    O=C1C=2C(=CC=C(C2)C=3C=NNC3)C=NN1CC4=CC(OC)=CC=C4

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound