GRK2i - CAS 148505-03-7

GRK2 inhibitory polypeptide that specifically inhibits Gβγ activation of GRK2. Corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist.

GRK

GPCR/G Protein

148505-03-7

C153H256N50O41S

3484.08

C([C@@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CC1=CC=C(O)C=C1)C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(=O)N2[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(=O)N3[C@H](C(N[C@H](C(N[C@H](C(O)=O)CO)=O)CCCNC(=N)N)=O)CCC3)CCCCN)=O)CC(N)=O)=O)CCCCN)=O)CCSC)=O)CCCCN)=O)CCC2)[C@H](C)C)=O)CCCNC(=N)N)=O)CCC(N)=O)=O)[C@H](C)C)=O)CC(C)C)=O)CCC(N)=O)=O)CCC(N)=O)=O)C)=O)CCC(O)=O)=O)CCCNC(=N)N)=O)=O)C)=O)CC(O)=O)=O)CCCNC(=N)N)=O)CC(C)C)=O)CCC(O)=O)=O)CCCCN)=O)CCCCN)=O)N)C=4C=5C(NC4)=CC=CC5

-20°C

Ice Packs

Peptide