1 1

Molfinity

GRP78-IN-3 - CAS 2707510-30-1

GRP78-IN-3 - CAS 2707510-30-1

MF-0098184-01

$42.89 USD
$42.89 USD
Sale Sold out
Taxes included.
Size
View full details

Product Details

  • Bioactivity

    GRP78-IN-3, a potent small-molecule-competitive inhibitor of Hsp70 substrate binding and is a selective Grp78 (HSPA5) inhibitor with an IC50 of 0.59 μM. GRP78-IN-3 is 7-fold selective for HspA5 compared to HspA9 (IC50 of 4.3 μM) and >20-fold selective for HspA5 compared to HspA2 (IC50 of 13.9 μM) .

  • Target

    HSP

  • Related Pathways

    Metabolism, Cytoskeletal Signaling

  • CAS Number

    2707479

  • Purity

    0.9949

  • Molecular Formula

    C17H18N4O2S

  • Molecular Weight

    342.42

  • SMILES

    C(N[C@H](C(NC1=NC=CS1)=O)[C@H](C)C)(=O)C2=CC=3C(N2)=CC=CC3

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound