GSK040 - CAS 2752331-09-0

GSK040, a potent and highly selective inhibitor of BET BD2, exhibits a pIC50 of 8.3, demonstrating over 5000-fold selectivity against BET BD1 (pIC50=4.6) . This compound is primarily utilized in oncology and immunology research [1].This compound is unstable in powder form and other related salt forms are recommended.

Epigenetic Reader Domain, Others

Chromatin/Epigenetic, Others

2752331-09-0

C29H34N4O4

502.6

N([C@@H](C(NC)=O)[C@@H]1CCOCC1)(C(=O)C=2C=C(C)C(=O)N(C)C2)C[C@H](C3=CC=CC=C3)C4=CC=CC=N4

-20°C

Ice Packs

Small Compound