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Molfinity

GSK046 - CAS 2474876-09-8

GSK046 - CAS 2474876-09-8

MF-0018666-01

$51.11 USD
$51.11 USD
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Product Details

  • Bioactivity

    GSK046 (iBET-BD2) is a potent, selective, and orally active BD2 bromodomain inhibitor of the BET proteins, with IC50 values of 264 nM [BRD2 BD2], 98 nM [BRD3 BD2], 49 nM [BRD4 BD2], and 214 nM [BRDT BD2], respectively. It exhibits immunomodulatory activity.

  • Target

    Epigenetic Reader Domain

  • Related Pathways

    Chromatin/Epigenetic

  • CAS Number

    2474876-09-8

  • Purity

    0.9997

  • Molecular Formula

    C23H27FN2O4

  • Molecular Weight

    414.47

  • SMILES

    C[C@H](Oc1cc(cc(F)c1NC(C)=O)C(=O)N[C@H]1CC[C@H](O)CC1)c1ccccc1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound