GSK172981 - CAS 1133705-99-3

GSK172981 is a non-peptide tachykinin NK3 receptor antagonist with a high affinity for the recombinant human (PK (I) value 7.7) and native guinea pig (PK (I) value 7.8) tachykinin NK3 receptor. In vitro, the functional evaluation showed that GSK172981 was a competitive antagonist for the cloned human tachykinin NK (3) receptor (PA (2) =7.2) . GSK172981 may be used to treat schizophrenia.

Others

Others

1133603

C26H22FN3O

411.47

C(N[C@@H]([C@@H]1CC1)C2=CC=CC=C2)(=O)C=3C4=C(N=C(C3N)C5=CC(F)=CC=C5)C=CC=C4

-20°C

Ice Packs

Small Compound