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Molfinity

GSK215 - CAS 2743427-26-9

GSK215 - CAS 2743427-26-9

MF-0098173-01

$128.19 USD
$128.19 USD
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Product Details

  • Bioactivity

    GSK215 is a potent and selective PROTAC focal adhesion kinase (FAK) degrader (pDC50= 8.4), designed using the FAK inhibitor VS-4718 and a binder for the VHL E3 ligase, capable of inducing rapid and prolonged FAK degradation.

  • Target

    PROTACs, FAK

  • Related Pathways

    Cytoskeletal Signaling, PROTAC, Tyrosine Kinase/Adaptors, Angiogenesis

  • CAS Number

    2743392

  • Purity

    0.993

  • Molecular Formula

    C50H59F3N10O6S

  • Molecular Weight

    985.13

  • SMILES

    CNC(=O)c1ccccc1Nc1cc(Nc2ccc(cc2OC)N2CCN(CC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(cc3)-c3scnc3C)C(C)(C)C)CC2)ncc1C(F)(F)F

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    PROTAC