HDAC8/BRPF1-IN-1 - CAS 2484255-85-6

HDAC8/BRPF1-IN-1 (Compound 23a) is a dual inhibitor targeting human HDAC8 (IC50: 443 nM) and human BRPF1 (Kd: 67 nM), with low in vitro activity against HDAC1 and HDAC6.

HDAC, Others, Epigenetic Reader Domain

Others, DNA Damage/DNA Repair, Chromatin/Epigenetic

2484164

C19H19N3O6S

417.44

CN1C=2C(=CC(NS(=O)(=O)C3=C(OC)C=CC(C(NO)=O)=C3)=CC2)C=C(C)C1=O

-20°C

Ice Packs

Small Compound