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KDM5A-IN-1 - CAS 1905481-36-8

KDM5A-IN-1 - CAS 1905481-36-8

SKU:MF-0015153-01

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  • Bioactivity

    KDM5A-IN-1 is an orally available, potent and selective inhibitor of the pan-histidine lysine demethylase 5 KDM5, inhibiting KDM5A, KDM5B, and KDM5C with IC50 values of 45 nM, 56 nM, and 55 nM, respectively.KDM5A-IN-1 inhibits PC9 H3K4Me3, and may be useful in cancer research.

  • Target

    Histone Demethylase

  • Related Pathways

    Chromatin/Epigenetic

  • CAS Number

    1905437

  • Purity

    >99.99%

  • Molecular Formula

    C15H22N4O2

  • Molecular Weight

    290.36

  • SMILES

    CC(C)c1cc([nH]n1)C(=O)N1CC[C@H](C1)NC(=O)C1CC1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound