Liarozole - CAS 115575-11-6

Liarozole (R75251 dihydrochloride) is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase) .Liarozole dihydrochloride is an imidazole derivative; it is being investigated as a non-hormonal agent in prostate cancer and in the treatment of various other cancers and skin disorders.

Cytochromes P450, Retinoid Receptor

Metabolism

115558

0.9938

C17H13ClN4

308.76

Clc1cccc(c1)C(c1ccc2nc[nH]c2c1)n1ccnc1

-20°C

Ice Packs

Small Compound