Linopirdine - CAS 105431-72-9

Linopirdine (DuP 996) is a TRPV1 agonist. Linopirdine is an orally active and selective M-type K+ current (IM; Kv7; KCNQ Channels) inhibitor (IC50: 2.4 μM) . Linopirdine is a cognitive enhancer. It acts by stimulating release of acetylcholine and other neurotransmitters.Linopirdine is a putative cognition-enhancing drug that increases acetylcholine release in rat brain tissue.

Potassium Channel, TRP/TRPV Channel

Membrane transporter/Ion channel

105350

0.9992

C26H21N3O

391.46

O=C1N(c2ccccc2C1(Cc1ccncc1)Cc1ccncc1)c1ccccc1

-20°C

Ice Packs

Small Compound