Lumateperone Tosylate - CAS 1187020-80-9

Lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist (Ki: 0.54 nM), a SERT blocker (Ki: 61 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki: 32 nM) .

5-HT Receptor, Dopamine Receptor

Neuroscience, GPCR/G Protein

1187020-80-9

0.9995

C31H36FN3O4S

565.7

Cc1ccc(cc1)S(O)(=O)=O.CN1CCN2C3CCN(CCCC(=O)c4ccc(F)cc4)CC3c3cccc1c23

-20°C

Ice Packs

Small Compound