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Molfinity

Lurosetron - CAS 128486-54-4

Lurosetron - CAS 128486-54-4

MF-0147962-01

$1,647.05 USD
$1,647.05 USD
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Product Details

  • Bioactivity

    Lurosetron (GR-87442) is the 6-fluoro analogue of Alosetron. It functions as a serotonin 5-HT3 receptor antagonist. Lurosetron inhibits recombinant (rbt) CYP1A2 with an IC50 of 0.1 μM and also inhibits other CYP subtypes, including rbtCYP2C9 and rbtCYP3A4, with IC50 values ranging from 3.5 μM to 16 μM.

  • Target

    5-HT Receptor

  • Related Pathways

    GPCR/G Protein, Neuroscience

  • CAS Number

    128486-54-4

  • Molecular Formula

    C17H17FN4O

  • Molecular Weight

    312.34

  • SMILES

    O=C1C=2C=3C=CC=C(F)C3N(C2CCN1CC=4NC=NC4C)C

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound