Lys-[Des-Arg9]Bradykinin TFA - CAS 2763588-90-3

Lys-[Des-Arg9]Bradykinin TFA is a naturally occurring kinin that serves as a potent and highly selective agonist for the bradykinin B1 receptor, demonstrating binding affinities (K i values) of 0.12 nM, 1.7 nM, and 0.23 nM for the human, mouse, and rabbit B1 receptors, respectively. This compound exhibits low inhibitory activity on B2 receptors [1] [2].

Bradykinin Receptor

GPCR/G Protein

2763495

C54H75F6N13O15

1260.24

OC(C(F)(F)F)=O.O=C(N1[C@@H](CCC1)C(NCC(N[C@H](C(N[C@@H](CO)C(N2[C@@H](CCC2)C(N[C@H](C(O)=O)CC3=CC=CC=C3)=O)=O)=O)CC4=CC=CC=C4)=O)=O)[C@H]5N(CCC5)C([C@H](CCCNC(N)=N)NC([C@@H](N)CCCCN)=O)=O.OC(C(F)(F)F)=O

-20°C

Ice Packs

Peptide