[Lys5, MeLeu9, Nle10]-NKA (4-10) - CAS 137565-28-7

Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM) . Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively) .

Neurokinin receptor

GPCR/G Protein, Neuroscience

137530

>99.99%

C39H65N9O9

803.99

[C@@H](CC1=CC=CC=C1)(NC([C@@H](NC([C@H](CC(O)=O)N)=O)CCCCN)=O)C(N[C@H](C(NCC(N([C@H](C(N[C@@H](CCCC)C(N)=O)=O)CC(C)C)C)=O)=O)C(C)C)=O

-20°C

Ice Packs

Peptide