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Molfinity

Mardepodect - CAS 898562-94-2

Mardepodect - CAS 898562-94-2

MF-0033769-01

$36.91 USD
$36.91 USD
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Product Details

  • Bioactivity

    Mardepodect (PF-2545920) is a phosphodiesterase inhibitor selective for the PDE10A subtype with an IC50 of 0.37 nM and over 1000-fold selectivity over PDE. It is potentially useful for the treatment of schizophrenia. Phosphodiesterase 10A (PDE10A) is highly expressed in striatal medium spiny neurons of both the direct and indirect output pathways. Mardepodect can cross the blood-brain barrier.

  • Target

    PDE

  • Related Pathways

    Metabolism

  • CAS Number

    898466

  • Purity

    0.9994

  • Molecular Formula

    C25H20N4O

  • Molecular Weight

    392.45

  • SMILES

    Cn1cc(c(n1)-c1ccc(OCc2ccc3ccccc3n2)cc1)-c1ccncc1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound