Masupirdine free base - CAS 701205-60-9

Masupirdine free base (SUVN-502 free base) is an orally available 5-HT6 receptor antagonist that crosses the blood-brain barrier, with a Ki value of 2.04 nM for the human 5-HT6 receptor. It is potent and selective, inhibiting multiple targets, and can be used in the study of neurological disorders such as Alzheimer's disease.

5-HT Receptor

GPCR/G Protein, Neuroscience

701136

0.9965

C21H24BrN3O3S

478.4

O=S(=O)(C=1C=CC=CC1Br)N2C=C(C=3C=C(OC)C=CC32)CN4CCN(C)CC4

-20°C

Ice Packs

Small Compound