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Molfinity

MDR-652 - CAS 1933528-96-1

MDR-652 - CAS 1933528-96-1

SKU:MF-0014900-01

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  • Bioactivity

    MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1), with Ki values of 11.4 nM and 23.8 nM for hTRPV1 and rTRPV1, respectively, and EC50s of 5.05 nM and 93 nM for hTRPV1 and rTRPV1, respectively. MDR-652 is a potent topical analgesic.

  • Target

    TRP/TRPV Channel

  • Related Pathways

    Membrane transporter/Ion channel

  • CAS Number

    1933431

  • Purity

    0.9996

  • Molecular Formula

    C22H23ClFN3O2S

  • Molecular Weight

    447.95

  • SMILES

    CC(C)(C)c1nc(c(CNC(=O)Nc2ccc(CO)c(F)c2)s1)-c1cccc(Cl)c1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound