Mirogabalin besylate - CAS 1138245-21-2

Mirogabalin besylate is a potent and orally active ligand that selectively targets the α2δ subunit of voltage-gated calcium channels. It displays high affinity (K d) values, namely 13.5 nM, 22.7 nM, 27 nM, and 47.6 nM, for human α2δ-1, human α2δ-2, rat α2δ-1, and rat α2δ-2, respectively.

Others, Calcium Channel

Metabolism, Others, Membrane transporter/Ion channel

1138245-21-2

C18H25NO5S

367.46

OS(=O)(=O)c1ccccc1.[H][C@@]12C[C@](CN)(CC(O)=O)[C@]1([H])C=C(CC)C2

-20°C

Ice Packs

Small Compound