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Molfinity

ML221 - CAS 877636-42-5

ML221 - CAS 877636-42-5

MF-0093233-01

$32.42 USD
$32.42 USD
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Product Details

  • Bioactivity

    ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the β-arrestin assay, and EC80 of 10 nM in both assays.

  • Target

    Arrestin, Apelin receptor

  • Related Pathways

    GPCR/G Protein

  • CAS Number

    877589

  • Purity

    0.9774

  • Molecular Formula

    C17H11N3O6S

  • Molecular Weight

    385.35

  • SMILES

    [O-][N+](=O)c1ccc(cc1)C(=O)Oc1coc(CSc2ncccn2)cc1=O

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound