ML252 - CAS 1392494-64-2

ML252 is a selective potassium channel inhibitor, specifically targeting the KCNQ2 channel (Kv7.2) with an IC50 value of 69 nM. Additionally, ML252 demonstrates inhibitory activity against Cytochrome P450 isoforms, including IC50 values of 6.1 nM (CYP1A2), 18.9 nM (CYP2C9), 3.9 nM (CYP3A4), and 19.9 nM (CYP2D6) .

Others, Potassium Channel, Cytochromes P450

Membrane transporter/Ion channel, Others, Metabolism

1392428

C20H24N2O

308.42

N(C([C@@H](CC)C1=CC=CC=C1)=O)C2=C(C=CC=C2)N3CCCC3

-20°C

Ice Packs

Small Compound