MRS2279 diammonium - CAS 2387505-47-5

MRS2279 diammonium, a selective and high-affinity P2Y1 receptor antagonist, exhibits a Ki value of 2.5 nM and an IC50 value of 51.6 nM. It competitively inhibits ADP-promoted platelet aggregation, demonstrating a pKb value of 8.05.

P2Y Receptor, Others

Neuroscience, GPCR/G Protein, Others

2387453

C13H24ClN7O8P2

503.77

C(OP(=O)(O)O)[C@]12[C@](C1)([C@H](C[C@@H]2OP(=O)(O)O)N3C=4C(N=C3)=C(NC)N=C(Cl)N4)[H].N

-20°C

Ice Packs

Small Compound