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Muscarinic toxin 3 - CAS 873336-87-9
Muscarinic toxin 3 - CAS 873336-87-9
SKU:MF-0158027-01
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Product Details
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Bioactivity
Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57 for α1B, 8.13 for α1D, 8.49 for α2A, <6.5 for α2B, and 7.29 for α2C receptors. MT3 notably demonstrates significant adrenoceptor activity [1].
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Target
AChR, Adrenergic Receptor
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Related Pathways
Neuroscience, GPCR/G Protein
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CAS Number
873240
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Molecular Formula
C319H489N89O97S8
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Molecular Weight
7379.35
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Storage Temperature
-20°C
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Shipping Conditions
Ice Packs
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Category
Peptide