N-Methylcytisine - CAS 486-86-2

1. N-Methylcytisine (Caulophylline) 's nicotinic receptors have high affinity (KD = 5 nM) to nAChR from squid optical ganglia. 2. N-Methylcytisine and N, N-dimethylcytisine did not displace 14C-tubocurarine at a concentration of .1 mM, cytisine was the only effective inhibitor of 14C-tubocurarine specific binding (Ki=7 nM) .

AChR

Neuroscience

398

0.9989

C12H16N2O

204.27

CN1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2

-20°C

Ice Packs

Natural Product