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αO-Conotoxin GeXIVA - CAS 2010167-25-4
αO-Conotoxin GeXIVA - CAS 2010167-25-4
SKU:MF-0158029-01
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Product Details
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Bioactivity
αO-Conotoxin GeXIVA, a potent antagonist of the α9α10 nicotinic acetylcholine receptor (nAChR), exhibits an inhibition concentration 50 (IC50) of 12 nM against rat α9α10 nAChRs. This compound has demonstrated analgesic properties in animal pain models [1].
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Target
AChR
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Related Pathways
Neuroscience
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CAS Number
2010138
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Molecular Formula
C139H227N55O41S4
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Molecular Weight
3452.89
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Storage Temperature
-20°C
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Shipping Conditions
Ice Packs
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Category
Peptide