P-gp/BCRP-IN-1 - CAS 2764596-06-5

P-gp/BCRP-IN-1 (compound 19) is a relatively safe, orally active, and efficient inhibitor of the efflux transporters P-gp and BCRP, which reverses resistance and enhances the oral bioavailability of Paclitaxel (PTX) [1].

BCRP, Others

Membrane transporter/Ion channel, Others

2764596-06-5

C27H25ClN4O3

488.97

C(NC1=CC=C(CCN2CCOCC2)C=C1)(=O)C=3C=4C(C(=O)N(N3)C5=CC=C(Cl)C=C5)=CC=CC4

-20°C

Ice Packs

Small Compound