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Molfinity

Pactimibe sulfate - CAS 608510-47-0

Pactimibe sulfate - CAS 608510-47-0

MF-0047514-01

$1,471.55 USD
$1,471.55 USD
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Product Details

  • Bioactivity

    Pactimibe sulfate (CS-505) is a dual ACAT1/2 inhibitor, acting on ACAT1 (IC50: 4.9 μM) and ACAT2 (IC50: 3.0 μM) . It inhibits oleoyl-CoA non-competitively (Ki: 5.6 μM) and significantly inhibits cholesterol ester formation (IC50: 6.7 μM) . Pactimibe sulfate reduces plasma cholesterol activity and has anti-atherogenic potential.

  • Target

    Others, Acyltransferase

  • Related Pathways

    Others, Metabolism

  • CAS Number

    608463

  • Molecular Formula

    C50H82N4O10S

  • Molecular Weight

    931.28

  • SMILES

    OS(O)(=O)=O.CCCCCCCCN1CCc2c1c(NC(=O)C(C)(C)C)c(C)c(CC(O)=O)c2C.CCCCCCCCN1CCc2c1c(NC(=O)C(C)(C)C)c(C)c(CC(O)=O)c2C

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound