Skip to product information
1 of 1

Molfinity

PBRM1-BD2-IN-1 - CAS 1915012-21-3

PBRM1-BD2-IN-1 - CAS 1915012-21-3

SKU:MF-0146385-01

Regular price $1,383.80 USD
Regular price Sale price $1,383.80 USD
Sale Sold out
Taxes included.
Size
Quantity
View full details
  • Bioactivity

    PBRM1-BD2-IN-1 is a selective and cell-active inhibitor of the polybromo-1 (PBRM1) bromodomain, exhibiting a binding affinity (Kd) of 0.7 μM and an inhibitory efficacy (IC50) of 0.2 μM, and is used in cancer research.

  • Target

    Others, Epigenetic Reader Domain

  • Related Pathways

    Chromatin/Epigenetic, Others

  • CAS Number

    1914988

  • Molecular Formula

    C17H19ClN2O

  • Molecular Weight

    302.8

  • SMILES

    C(\C(CC)CC)=C\1/C=2N(C=3C(C(=O)N2)=C(Cl)C=CC3)CC1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound