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Molfinity

PBRM1-BD2-IN-2 - CAS 2819989-57-4

PBRM1-BD2-IN-2 - CAS 2819989-57-4

SKU:MF-0012060-01

Regular price $120.06 USD
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  • Bioactivity

    PBRM1-BD2-IN-2, a selective and cell-active inhibitor of the polybromo-1 (PBRM1) bromodomain, exhibits binding affinity and inhibitory activity specifically targeting the PBRM1-BD2 domain, with Kd and IC50 values of 9.3 μM and 1.0 μM, respectively. This compound is utilized in cancer research.

  • Target

    Epigenetic Reader Domain

  • Related Pathways

    Chromatin/Epigenetic

  • CAS Number

    2819989-57-4

  • Purity

    >99.99%

  • Molecular Formula

    C14H9Cl2FN2O

  • Molecular Weight

    311.14

  • SMILES

    O=C1C=2C(NC(N1)C3=C(Cl)C=CC=C3F)=CC=CC2Cl

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound