PCS1055 - CAS 357173-55-8

PCS1055 is a selective and competitive antagonist of the muscarinic M4 receptor (muscarinic M4 receptor), with an IC50 of 18.1 nM and a Kd of 5.72 nM. It inhibits the binding of the radioligand [3H]-NMS to the M4 receptor, with a Ki of 6.5 nM. Additionally, PCS1055 acts as an AChE inhibitor, exhibiting IC50 values of 22 nM for electric eel AChE and 120 nM for human AChE.

AChR, Cholinesterase (ChE)

Neuroscience

357173-55-8

C27H32N4

412.57

N1=NC=2C3=CC=CC=C3CCCC2C=C1NCCC4CCN(CC=5C=CC=CC5)CC4

-20°C

Ice Packs

Small Compound