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PDE4B/7A-IN-2 - CAS 2511632-55-4

PDE4B/7A-IN-2 - CAS 2511632-55-4

MF-0050407-01

$1,383.80 USD
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Product Details

  • Bioactivity

    This compound is a dual 5-HT1A/5-HT7 receptor antagonist (5-HT1A Ki = 8 nM, Kb = 0.04 nM; 5-HT7 Ki = 451 nM, Kb = 460 nM) with additional inhibitory activity against PDE4B/PDE7A (PDE4B IC50 = 80.4 μM; PDE7A IC50 = 151.3 μM) . Its antidepressant-like effect surpasses that of the reference agent, escitalopram.

  • Target

    Others, PDE

  • Related Pathways

    Others, Metabolism

  • CAS Number

    2511573

  • Molecular Formula

    C25H35N3O2

  • Molecular Weight

    409.56

  • SMILES

    O(C)C1=C(C=CC=C1)N2CCN(CCCCC(NC3=CC=C(C(C)C)C=C3)=O)CC2

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound