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Molfinity

PF-4981517 - CAS 1390637-82-7

PF-4981517 - CAS 1390637-82-7

MF-0094330-01

$41.39 USD
$41.39 USD
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Product Details

  • Bioactivity

    PF-4981517 (CYP3cide) is a efficient, specific and time-dependent inhibitor of cytochrome P4503A4 (CYP3A4) . The IC 50 values for CYP3A activity are 0.03 μM,17 μM, and 71 μM for CYP3A4, CYP3A5, and CYP3A7, respectively. PF-4981517 is able to be used to distinguish the contributions of CYP3A4 versus CYP3A5 on drug Metabolism.

  • Target

    Cytochromes P450

  • Related Pathways

    Metabolism

  • CAS Number

    1390548

  • Purity

    0.9983

  • Molecular Formula

    C26H32N8

  • Molecular Weight

    456.59

  • SMILES

    Cc1ccc(cc1)-c1c(cnn1C)-c1nn(C)c2ncnc(N3CC[C@@H](C3)N3CCCCC3)c12

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound