PG106 - CAS 944111-22-2

Selective hMC3 receptor antagonist (IC50 = 210 nM) . Exhibits no activity at hMC4 receptors and hMC5 receptors.

Melanocortin Receptor

GPCR/G Protein, Neuroscience

944087

C51H69N13O9

1008.19

C(C=1C=2C(NC1)=CC=CC2)[C@@H]3NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](CC4=CC5=C(C=C4)C=CC=C5)NC(=O)CCNC(=O)[C@@H](NC([C@H](CCCC)NC(C)=O)=O)CC(=O)NCCCC[C@@H](C(N)=O)NC3=O

-20°C

Ice Packs

Peptide