[Phe1Ψ (CH2-NH) Gly2]Nociceptin (1-13) NH2 - CAS 213130-17-7

Potent agonist of the nociceptin (ORL1) receptor, demonstrated both in vitro and in vivo. Selective, competitive antagonism at the nociceptin receptor has also been reported (pA2 = 7.02 and 6.75 in the guinea pig ileum and mouse vas deferens respectively) .

Opioid Receptor

GPCR/G Protein, Endocrinology/Hormones, Neuroscience

213106

C61H102N22O14

1367.6

[C@H](CC1=CC=CC=C1)(C(N[C@H](C(NCC(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CCCCN)C(N)=O)=O)CCCNC(=N)N)=O)C)=O)CO)=O)CCCCN)=O)CCCNC(=N)N)=O)C)=O)=O)[C@@H](C)O)=O)NC(CNC(CNC[C@H](CC2=CC=CC=C2)N)=O)=O

-20°C

Ice Packs

Peptide