PKG inhibitor peptide - CAS 82801-73-8

Competitive inhibitor of cGMP-dependent protein kinase (PKG) ; analog of a substrate peptide corresponding to a phosphorylation site of histone H2B. Competes with synthetic substrates (Ki = 86 mM) but does not inhibit phosphorylation of intact histones by PKG. Inhibits phosphorylation of intact histones by PKA.

PKA

Tyrosine Kinase/Adaptors

82720

C38H74N18O10

943.12

C[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](N)CCCNC(N)=N)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(O)=O

-20°C

Ice Packs

Peptide