PKN3-IN-1 - CAS 2361545-75-5

PKN3-IN-1 (compound 16) inhibits PKN3 (serine/threonine-protein kinase N3) and GAK (cyclin G-associated kinase) with an IC50 of 0.014 μM and a Ki of 0.0044 μM. PKN3-IN-1 is a potential tool compound for investigating the cell biology of PKN3 and its role in pancreatic and prostate cancers, as well as T-cell acute lymphoblastic leukemia.

PI3K

PI3K/Akt/mTOR signaling

2361465

C18H17IN2O3

436.244

IC=1C=CC=2C(=NC=CC2NC3=CC(OC)=C(OC)C(OC)=C3)C1

-20°C

Ice Packs

Small Compound