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Molfinity

PKRA83 - CAS 1233926-87-8

PKRA83 - CAS 1233926-87-8

MF-0137865-01

$1,654.95 USD
$1,654.95 USD
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Product Details

  • Bioactivity

    PKRA83 is a potent prokineticin (PK2) antagonist that crosses the blood-brain barrier and competes for PK2 binding to its receptors PKR1 and PKR2. PKRA83 effectively inhibits PK2 receptors and acts on PKR1 (IC50: 5.0 nM) and PKR2 (IC50: 8.2 nM) . PKRA83 exhibits anti-cancer and anti-angiogenic effects.

  • Target

    Others

  • Related Pathways

    Others

  • CAS Number

    1233831

  • Molecular Formula

    C27H34ClFN2O4

  • Molecular Weight

    505.02

  • SMILES

    ClC1=C2C(=CC(CN(C(=O)[C@H]3CN(CC4=CC(OC)=C(F)C=C4)CC3)CC(C)C)=C1)OCCCO2

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound