PL-017 - CAS 83397-56-2

Selective μ opioid receptor agonist (IC50 values are 5.5 and > 10000 nM for inhibition of 125I-FK 33,824 and 125I-DADLE binding to μ and δ sites respectively) . Produces naloxone-reversible analgesia, catalepsy and hyperthermia following central administration in rats in vivo.

Opioid Receptor

GPCR/G Protein, Neuroscience, Endocrinology/Hormones

83339

C29H37N5O5

535.64

C(N([C@H](C(=O)N1[C@@H](C(N)=O)CCC1)CC2=CC=CC=C2)C)(=O)[C@H]3N(C([C@H](CC4=CC=C(O)C=C4)N)=O)CCC3

-20°C

Ice Packs

Peptide