PQM-244 - CAS 316139-50-1

PQM-244 (Compound 5c) is an orally active multi-target modulator that acts on TRPV1, CB1, and CB2 receptors. It exhibits significant peripheral analgesic effects during both neurogenic and inflammatory phases. PQM-244 also shows potential antioxidant activity with a DPPH radical scavenging IC50 of 14.15 μM. This compound is applicable for research into chronic pain and inflammatory diseases, such as diabetes, atherosclerosis, and Alzheimer's disease.

Cannabinoid Receptor, TRP/TRPV Channel

GPCR/G Protein, Membrane transporter/Ion channel

316088

C18H22N2O2

298.38

O=C(NN=C1C(=CCC(C(=C)C)C1)C)C2=CC=C(OC)C=C2

-20°C

Ice Packs

Small Compound