PSB-1901 free base - CAS 2332835-02-4

PSB-1901 is a potent A2B Adenosine Receptor Antagonist with Picomolar Potency (Ki 0.0835 nM, KB 0.0598 nM, human A2BAR) with >10 000-fold selectivity versus all other AR subtypes. PSB-1901 was similarly potent and selective at the mouse A2BAR, making it a promising tool for preclinical studies.

Adenosine Receptor, Others

Others, Neuroscience, GPCR/G Protein

2332835-02-4

C24H25BrN6O4S

573.46

O=C1C2=C(N=C(N2)C3=CC=C(S(=O)(=O)N4CCN(CC4)C5=CC=C(Br)C=C5)C=C3)NC(=O)N1CCC

-20°C

Ice Packs

Small Compound