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Molfinity

Pyr6 - CAS 245747-08-4

Pyr6 - CAS 245747-08-4

MF-0019114-01

$33.17 USD
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Product Details

  • Bioactivity

    Pyr6 (N-[4-[3,5-Bis (trifluoromethyl) -1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide) is a selective TRPC3 inhibitor with IC50 of 0.49 uM (Ca2+ influx inhibition in thapsigargin depleted native RBL-2H3 cells) .Pyr6 is an inhibitor of Ca2+ entry, which displays higher potency to inhibit Ca2+ entry mediated by CRAC channel than by TRPC3.

  • Target

    Calcium Channel, TRP/TRPV Channel

  • Related Pathways

    Metabolism, Membrane transporter/Ion channel

  • CAS Number

    245747-08-4

  • Purity

    0.9918

  • Molecular Formula

    C17H9F7N4O

  • Molecular Weight

    418.27

  • SMILES

    Fc1cnccc1C(=O)Nc1ccc(cc1)-n1nc(cc1C(F)(F)F)C(F)(F)F

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound