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(R) -GSK-3685032 - CAS 2170140-50-6

(R) -GSK-3685032 - CAS 2170140-50-6

MF-0006562-01

$337.82 USD
$213.20 USD $337.82 USD
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Product Details

  • Bioactivity

    (R) -GSK-3685032 is the R-enantiomer of GSK-3685032, a first-in-class, non-time-dependent, non-covalent, reversible, selective DNMT1 inhibitor with an IC50 of 0.036 μM, which induces robust loss of DNA methylation, transcriptional activation, and inhibition of cancer cell growth.

  • Target

    Others, DNA Methyltransferase

  • Related Pathways

    Chromatin/Epigenetic, Others

  • CAS Number

    2170140-50-6

  • Molecular Formula

    C22H24N6OS

  • Molecular Weight

    420.54

  • SMILES

    CCc1c(C#N)c(S[C@@H](C(N)=O)c2ccccc2)nc(N2CCC(N)CC2)c1C#N

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound