(R) -YNT-3708 - CAS 2923137-94-2

(R) -YNT-3708 is a specific Orexin 1 receptor (OX1R) agonist with an EC50 value of 7.48 nM for OX1R. The EC50 ratio of OX2R to OX1R is 22.5. This compound demonstrates analgesic and enhancing effects by activating OX1R in mice.

OX Receptor

GPCR/G Protein, Neuroscience

2923041

C35H36N4O6S

640.75

N(C(CC1=CC(OC)=CC=C1)=O)(C)[C@H]2C=3C(=CC=C(NS(=O)(=O)C4=C(OC)C=CC(/C=C/C(NC=5C=CN=CC5)=O)=C4)C3)CCC2

-20°C

Ice Packs

Small Compound