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Molfinity

Relutrigine - CAS 2392951-29-8

Relutrigine - CAS 2392951-29-8

MF-0095267-01

$303.60 USD
$303.60 USD
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Product Details

  • Bioactivity

    Relutrigine (PRAX-562) is an orally active, long-acting sodium current inhibitor that preferentially suppresses sustained INa induced by TX-II or SCN8A N1768D mutations (IC50=141/75 nM) . It reduces neuronal intrinsic excitability and may be used for anticonvulsant therapy.

  • Target

    Sodium Channel

  • Related Pathways

    Membrane transporter/Ion channel

  • CAS Number

    2392914

  • Purity

    0.9968

  • Molecular Formula

    C15H11F6N5O2

  • Molecular Weight

    407.27

  • SMILES

    C(OCC)(F)(F)C=1N2C(=NN1)C=NC(=C2)C=3C=C(F)C(OCC(F)(F)F)=NC3

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound