RS-102221 - CAS 185376-97-0

RS-102221 is a selective antagonist of the 5-HT2C receptor with a K i of 10 nM, demonstrating nearly 100-fold more selectivity for the 5-HT2C receptor over the 5-HT2A and 5-HT2B receptors. This compound not only has the potential to promote the differentiation of new nerve cells but also increases food intake and weight gain in rats.

5-HT Receptor

GPCR/G Protein, Neuroscience

185279

C27H31F3N4O7S

612.62

O=C1NC(=O)C2(N1)CCN(CCCCC(=O)C3=CC(NS(=O)(=O)C4=CC=C(C=C4)C(F)(F)F)=C(OC)C=C3OC)CC2

-20°C

Ice Packs

Small Compound